Inventors:
Xiangping Qian - South San Francisco CA, US
Andrew McDonald - San Francisco CA, US
Han-Jie Zhou - South San Francisco CA, US
Luke Ashcraft - South San Francisco CA, US
Bing Yao - South San Francisco CA, US
Hong Jiang - South San Francisco CA, US
Jennifer Kuo Chen Huang - South San Francisco CA, US
Jianchao Wang - South San Francisco CA, US
David Morgans - South San Francisco CA, US
Bradley Morgan - South San Francisco CA, US
Gustave Bergnes - South San Francisco CA, US
Dashyant Dhanak - Philadelphia PA, US
Steven Knight - Philadelphia PA, US
Nicholas Adams - Philadelphia PA, US
Cynthia Parrish - Philadelphia PA, US
Kevin Duffy - Philadelphia PA, US
Duke Fitch - Philadelphia PA, US
Rosanna Tedesco - Philadelphia PA, US
International Classification:
A61K 31/4184, A61K 31/4172, C07D 233/61
US Classification:
514394000, 514400000, 514614000, 548304400, 548335500, 564050000
Abstract:
Compounds useful for treating cellular proliferative diseases and disorders by modulating the activity of one or more mitotic kinesins are disclosed.